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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Sodium/potassium-transporting ATPase subunit alpha-2/beta-3
(Homo sapiens (Human))
Yeda Research and Development
US Patent
Ligand
BDBM444994
(US10668094, Compound DTMS-(silyl))
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Affinity Data
Ki: 11.1nM
Assay Description:
To screen for isoform selectivity of the digoxin derivatives we compared inhibition of Na,K-ATPase activity of purified detergent-soluble human isofo...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Sodium/potassium-transporting ATPase subunit alpha-2/beta-2
(Homo sapiens (Human))
Yeda Research and Development
US Patent
Ligand
BDBM444994
(US10668094, Compound DTMS-(silyl))
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Affinity Data
Ki: 14.3nM
Assay Description:
To screen for isoform selectivity of the digoxin derivatives we compared inhibition of Na,K-ATPase activity of purified detergent-soluble human isofo...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Sodium/potassium-transporting ATPase subunit alpha-2/beta-1
(Homo sapiens (Human))
Yeda Research and Development
US Patent
Ligand
BDBM444994
(US10668094, Compound DTMS-(silyl))
Copy SMILES
Copy InChI
Affinity Data
Ki: 24.3nM
Assay Description:
To screen for isoform selectivity of the digoxin derivatives we compared inhibition of Na,K-ATPase activity of purified detergent-soluble human isofo...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Sodium/potassium-transporting ATPase subunit alpha-1/beta-1
(Homo sapiens (Human))
Yeda Research and Development
US Patent
Ligand
BDBM444994
(US10668094, Compound DTMS-(silyl))
Copy SMILES
Copy InChI
Affinity Data
Ki: 72.6nM
Assay Description:
To screen for isoform selectivity of the digoxin derivatives we compared inhibition of Na,K-ATPase activity of purified detergent-soluble human isofo...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI