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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
24
hits in this display
Target
TGF-beta receptor type-1
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 42.2nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ3 family of Ser/Thr kinases. The kinases ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
TGF-beta receptor type-1
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 42.2nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
TGF-beta receptor type-1
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 42.2nM
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
TGF-beta receptor type-1
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 42.2nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Activin receptor type-1B
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 114nM
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Activin receptor type-1B
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 114nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Activin receptor type-1B
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 114nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Activin receptor type-1B
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 114nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ3 family of Ser/Thr kinases. The kinases ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Serine/threonine-protein kinase receptor R3
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 7.30E+3nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ3 family of Ser/Thr kinases. The kinases ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Serine/threonine-protein kinase receptor R3
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 7.30E+3nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Serine/threonine-protein kinase receptor R3
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 7.30E+3nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Serine/threonine-protein kinase receptor R3
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 7.30E+3nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Bone morphogenetic protein receptor type-1A
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+6nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ3 family of Ser/Thr kinases. The kinases ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Activin receptor type-1
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+6nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ3 family of Ser/Thr kinases. The kinases ...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Bone morphogenetic protein 10
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+6nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Bone morphogenetic protein receptor type-1A
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+6nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Activin receptor type-1
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+6nM
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Bone morphogenetic protein receptor type-1B
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+6nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Bone morphogenetic protein receptor type-1A
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+6nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Activin receptor type-1
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+6nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Bone morphogenetic protein receptor type-1B
(Mouse)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+6nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Bone morphogenetic protein receptor type-1A
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+6nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Bone morphogenetic protein receptor type-1B
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+6nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ3 family of Ser/Thr kinases. The kinases ...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Activin receptor type-1
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280349
((S)-4-(2-(5-chloro-2-fluorophenyl)-5-(dimethylamin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+6nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI