Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetRetinoic acid receptor RXR-alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290186((2E,4E)-3-Methyl-5-[(1R,2R)-1-methyl-2-(5,5,8,8-te...)
Affinity DataKi:  4nMAssay Description:Inhibition of [3H]-9-cis-RA binding to Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor RXR-gamma(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50290186((2E,4E)-3-Methyl-5-[(1R,2R)-1-methyl-2-(5,5,8,8-te...)
Affinity DataKi:  7nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor RXR-beta(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50290186((2E,4E)-3-Methyl-5-[(1R,2R)-1-methyl-2-(5,5,8,8-te...)
Affinity DataKi:  10nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290186((2E,4E)-3-Methyl-5-[(1R,2R)-1-methyl-2-(5,5,8,8-te...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ATRA binding to retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor beta(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290186((2E,4E)-3-Methyl-5-[(1R,2R)-1-methyl-2-(5,5,8,8-te...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ATRA binding to retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290186((2E,4E)-3-Methyl-5-[(1R,2R)-1-methyl-2-(5,5,8,8-te...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ATRA binding to Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor RXR-gamma(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50290186((2E,4E)-3-Methyl-5-[(1R,2R)-1-methyl-2-(5,5,8,8-te...)
Affinity DataEC50:  16nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290186((2E,4E)-3-Methyl-5-[(1R,2R)-1-methyl-2-(5,5,8,8-te...)
Affinity DataEC50:  1.78E+3nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor RXR-beta(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50290186((2E,4E)-3-Methyl-5-[(1R,2R)-1-methyl-2-(5,5,8,8-te...)
Affinity DataEC50:  14nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor RXR-alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290186((2E,4E)-3-Methyl-5-[(1R,2R)-1-methyl-2-(5,5,8,8-te...)
Affinity DataEC50:  7nMAssay Description:Inhibition of [3H]-9-cis-RA binding to Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor beta(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290186((2E,4E)-3-Methyl-5-[(1R,2R)-1-methyl-2-(5,5,8,8-te...)
Affinity DataEC50:  809nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails Article