Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179124((R,2E,4E)-3-methyl-5-(1-(5,5,8,8-tetramethyl-5,6,7...)
Affinity DataKi:  103nMAssay Description:Binding affinity to RXRalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-beta(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179124((R,2E,4E)-3-methyl-5-(1-(5,5,8,8-tetramethyl-5,6,7...)
Affinity DataKi:  188nMAssay Description:Binding affinity to RXRbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-gamma(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179124((R,2E,4E)-3-methyl-5-(1-(5,5,8,8-tetramethyl-5,6,7...)
Affinity DataKi:  202nMAssay Description:Binding affinity to RXRgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-beta(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179124((R,2E,4E)-3-methyl-5-(1-(5,5,8,8-tetramethyl-5,6,7...)
Affinity DataEC50:  1.29E+3nMAssay Description:Transactivation of RXRbeta in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-gamma(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179124((R,2E,4E)-3-methyl-5-(1-(5,5,8,8-tetramethyl-5,6,7...)
Affinity DataEC50:  1.26E+3nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed