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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
24
hits in this display
Target
TGF-beta receptor type-1
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 77.3nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ3 family of Ser/Thr kinases. The kinases ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
TGF-beta receptor type-1
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 77.3nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
TGF-beta receptor type-1
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 77.3nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
TGF-beta receptor type-1
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 77.3nM
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Activin receptor type-1B
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 149nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ3 family of Ser/Thr kinases. The kinases ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Activin receptor type-1B
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 149nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Activin receptor type-1B
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 149nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Activin receptor type-1B
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 149nM
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Serine/threonine-protein kinase receptor R3
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Activin receptor type-1
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Bone morphogenetic protein receptor type-1A
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Bone morphogenetic protein 10
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Serine/threonine-protein kinase receptor R3
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ3 family of Ser/Thr kinases. The kinases ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Activin receptor type-1
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ3 family of Ser/Thr kinases. The kinases ...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Bone morphogenetic protein receptor type-1A
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ3 family of Ser/Thr kinases. The kinases ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Bone morphogenetic protein receptor type-1B
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Bone morphogenetic protein receptor type-1A
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Activin receptor type-1
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Serine/threonine-protein kinase receptor R3
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Bone morphogenetic protein receptor type-1B
(Mouse)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Bone morphogenetic protein receptor type-1A
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Bone morphogenetic protein receptor type-1B
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ3 family of Ser/Thr kinases. The kinases ...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Serine/threonine-protein kinase receptor R3
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Activin receptor type-1
(Human)
Medivation Technologies
US Patent
Ligand
BDBM280368
(2-(5-chloro-2-fluorophenyl)-5-(prop-1-en-2-yl)-N-[...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Compound of the invention were screened in an in vitro kinase assay against several members of the TGFβ family of Ser/Thr kinases. The kinases t...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI