Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetThyrotropin receptor(Human)
Byondis

Curated by ChEMBL
LigandPNGBDBM50614114(CHEMBL5268512)
Affinity DataIC50:  91nMAssay Description:Antagonist activity at human TSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetThyrotropin receptor(Rat)
Byondis

Curated by ChEMBL
LigandPNGBDBM50614114(CHEMBL5268512)
Affinity DataIC50:  187nMAssay Description:Antagonist activity at TSHR in rat FRTL-5 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Human)
Byondis

Curated by ChEMBL
LigandPNGBDBM50614114(CHEMBL5268512)
Affinity DataIC50:  5.67E+3nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed