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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
NACHT, LRR and PYD domains-containing protein 3
(Human)
The Noguchi Institute
Curated by
ChEMBL
Ligand
BDBM50276372
(CHEMBL4128176)
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Affinity Data
IC50: 4.30E+3nM
Assay Description:
Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
NACHT, LRR and PYD domains-containing protein 3
(Mouse)
The Noguchi Institute
Curated by
ChEMBL
Ligand
BDBM50276372
(CHEMBL4128176)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5.70E+3nM
Assay Description:
Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI