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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
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Target
Proteasome subunit beta type-5
(Human)
Guangzhou Medical University
Curated by
ChEMBL
Ligand
BDBM50593023
(CHEMBL5183504)
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Affinity Data
IC50: 1.10nM
Assay Description:
Inhibition of 20S proteasome beta5 subunit (unknown origin) using Suc-LLVY-AMC as flurogenic substrate measured after 1 hr by fluorescence based anal...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
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Target
NACHT, LRR and PYD domains-containing protein 3
(Mouse)
Guangzhou Medical University
Curated by
ChEMBL
Ligand
BDBM50593023
(CHEMBL5183504)
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Copy InChI
Affinity Data
IC50: 49nM
Assay Description:
Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI