Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 9 hits in this display
BDBM579522(US11484525, Compound DD-63L-LB-S)
BDBM579520(US11484525, Compound DD-63L-LA-R | US11484525, Com...)Ki: 14nMAssay Description:Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...More data for this Ligand-Target Pair
BDBM579520(US11484525, Compound DD-63L-LA-R | US11484525, Com...)
Ki: 19nMAssay Description:Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...More data for this Ligand-Target Pair
BDBM579522(US11484525, Compound DD-63L-LB-S)
Ki: 22nMAssay Description:Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...More data for this Ligand-Target Pair
BDBM579520(US11484525, Compound DD-63L-LA-R | US11484525, Com...)
Ki: 43nMAssay Description:Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...More data for this Ligand-Target Pair
BDBM579520(US11484525, Compound DD-63L-LA-R | US11484525, Com...)
Ki: 44nMAssay Description:Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...More data for this Ligand-Target Pair
BDBM579520(US11484525, Compound DD-63L-LA-R | US11484525, Com...)
Ki: 67nMAssay Description:Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...More data for this Ligand-Target Pair
BDBM579520(US11484525, Compound DD-63L-LA-R | US11484525, Com...)
Ki: 83nMAssay Description:Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...More data for this Ligand-Target Pair
BDBM579522(US11484525, Compound DD-63L-LB-S)
Ki: 110nMAssay Description:Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...More data for this Ligand-Target Pair