Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetAlpha-2A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473619(CHEMBL130884)
Affinity DataKi:  91nMAssay Description:Displacement of [3H]RX821002 from human adrenergic alpha2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50473619(CHEMBL130884)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]clonidine from Alpha-2 adrenergic receptor of rat cortex membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473619(CHEMBL130884)
Affinity DataKi:  708nMAssay Description:Displacement of [3H]RX821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473619(CHEMBL130884)
Affinity DataKi:  1.15E+3nMAssay Description:Displacement of [3H]RX821002 from human adrenergic alpha-2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473619(CHEMBL130884)
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473619(CHEMBL130884)
Affinity DataEC50:  389nMAssay Description:Agonist activity at human adrenergic alpha-2A receptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473619(CHEMBL130884)
Affinity DataEC50:  93nMAssay Description:Agonist activity at human adrenergic alpha-2C receptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473619(CHEMBL130884)
Affinity DataEC50:  3.80E+3nMAssay Description:Agonist activity at human adrenergic alpha-2B receptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed