Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 40 hits in this display
BDBM50085683((+)-4-((S)-alpha,2,3-trimethylbenzyl)imidazole | 4...)
BDBM50085683((+)-4-((S)-alpha,2,3-trimethylbenzyl)imidazole | 4...)
BDBM50085683((+)-4-((S)-alpha,2,3-trimethylbenzyl)imidazole | 4...)
BDBM50085683((+)-4-((S)-alpha,2,3-trimethylbenzyl)imidazole | 4...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50085683((+)-4-((S)-alpha,2,3-trimethylbenzyl)imidazole | 4...)
Ki: 2.5nMAssay Description:Displacement of [3H]RS-79948-197 from recombinant human alpha2A adrenoreceptor expressed in CHOK1 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50085683((+)-4-((S)-alpha,2,3-trimethylbenzyl)imidazole | 4...)
BDBM50085683((+)-4-((S)-alpha,2,3-trimethylbenzyl)imidazole | 4...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50036913((+-)-4-(alpha,2,3-trimethylbenzyl)imidazole | 4-[1...)
BDBM50036913((+-)-4-(alpha,2,3-trimethylbenzyl)imidazole | 4-[1...)
BDBM50085683((+)-4-((S)-alpha,2,3-trimethylbenzyl)imidazole | 4...)
Ki: 31nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2c receptor expressed in CHO cells in presence of GppNHp/NaChecked by AuthorMore data for this Ligand-Target Pair
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
BDBM50036913((+-)-4-(alpha,2,3-trimethylbenzyl)imidazole | 4-[1...)
BDBM50036913((+-)-4-(alpha,2,3-trimethylbenzyl)imidazole | 4-[1...)
BDBM50036913((+-)-4-(alpha,2,3-trimethylbenzyl)imidazole | 4-[1...)
BDBM50036913((+-)-4-(alpha,2,3-trimethylbenzyl)imidazole | 4-[1...)
IC50: 3.40E+3nMAssay Description:Tested for its ability to antagonize epinephrine induced primary wave aggregation in human platelets at alpha-2A-adrenergic receptor sites.More data for this Ligand-Target Pair
BDBM50036913((+-)-4-(alpha,2,3-trimethylbenzyl)imidazole | 4-[1...)
BDBM50085683((+)-4-((S)-alpha,2,3-trimethylbenzyl)imidazole | 4...)
EC50: 2.10nMAssay Description:Agonist activity at recombinant human alpha2A adrenoreceptor expressed in CHOK1 cell membrane incubated for 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
BDBM50085683((+)-4-((S)-alpha,2,3-trimethylbenzyl)imidazole | 4...)