Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetKappa-type opioid receptor(Human)
The Regents of The University of California

US Patent
LigandPNGBDBM579515(US11484525, Compound DD-88B-S)
Affinity DataKi:  4.5nMAssay Description:Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetMu-type opioid receptor [N127C](Human)
The Regents of The University of California

US Patent
LigandPNGBDBM579515(US11484525, Compound DD-88B-S)
Affinity DataKi:  41nMAssay Description:Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetKappa-type opioid receptor(Human)
The Regents of The University of California

US Patent
LigandPNGBDBM579513(US11484525, Compound DD-88A-R)
Affinity DataKi:  60nMAssay Description:Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetMu-type opioid receptor [N127C](Human)
The Regents of The University of California

US Patent
LigandPNGBDBM579513(US11484525, Compound DD-88A-R)
Affinity DataKi:  96nMAssay Description:Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetDelta-type opioid receptor(Human)
The Regents of The University of California

US Patent
LigandPNGBDBM579513(US11484525, Compound DD-88A-R)
Affinity DataKi:  470nMAssay Description:Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetDelta-type opioid receptor(Human)
The Regents of The University of California

US Patent
LigandPNGBDBM579515(US11484525, Compound DD-88B-S)
Affinity DataKi:  570nMAssay Description:Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent