Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

LigandPNGBDBM50226961(CHEMBL38788)
Affinity DataKi:  0.960nMAssay Description:Inhibition of saturable binding of [3H]idazoxan to alpha2-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226961(CHEMBL38788)
Affinity DataKi:  1.90nMAssay Description:Binding affinity against alpha-2 adrenergic receptor was determined by the displacement of [3H]clonidine from rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Reckitt and Colman

Curated by ChEMBL
LigandPNGBDBM50226961(CHEMBL38788)
Affinity DataKi:  3.70nMAssay Description:Inhibition of saturable binding of [3H]prazosin to alpha1-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed