Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetRetinoic acid receptor beta(Human)
University of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50080526(1,4,4-Trimethyl-1,2,3,4-tetrahydro-quinoline-6-car...)
Affinity DataEC50:  256nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-gamma(Mouse)
University of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50080526(1,4,4-Trimethyl-1,2,3,4-tetrahydro-quinoline-6-car...)
Affinity DataEC50:  20nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-beta(Mouse)
University of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50080526(1,4,4-Trimethyl-1,2,3,4-tetrahydro-quinoline-6-car...)
Affinity DataEC50:  33nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Human)
University of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50080526(1,4,4-Trimethyl-1,2,3,4-tetrahydro-quinoline-6-car...)
Affinity DataEC50:  1.13E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed