Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetGTPase KRas [G12D](Homo sapiens (Human))
Shy Therapeutics

US Patent
LigandPNGBDBM485676(US10940139, Example 02903 | US11000515, Compound T...)
Affinity DataIC50:  2.05E+4nMAssay Description:Buffer-I: 50 mM Tris, pH 7.5 150 mM NaCl (optional) 1 mM MgCl2 1 mM DTT. KRas G12D mutant protein was expressed as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGTPase KRas [G12D,Q61H](Homo sapiens (Human))
Shy Therapeutics

US Patent
LigandPNGBDBM485676(US10940139, Example 02903 | US11000515, Compound T...)
Affinity DataIC50:  2.05E+4nMAssay Description:The following method was developed as specific assay for KRas G12D mutant protein.Buffer-I:50 mM Tris, pH 7.5150 mM NaCl (optional)1 mM MgCl21 mM DTT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGTPase KRas [G12D,Q61H](Homo sapiens (Human))
Shy Therapeutics

US Patent
LigandPNGBDBM485676(US10940139, Example 02903 | US11000515, Compound T...)
Affinity DataIC50:  2.05E+4nMAssay Description:The following method was developed as specific assay for KRas G12D mutant protein.Buffer-I: 50 mM Tris, pH 7.5 150 mM NaCl (optional) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGTPase KRas [G12D,Q61H](Homo sapiens (Human))
Shy Therapeutics

US Patent
LigandPNGBDBM485676(US10940139, Example 02903 | US11000515, Compound T...)
Affinity DataIC50:  2.05E+4nMAssay Description:Buffer-I: 50 mM Tris, pH 7.5 150 mM NaCl (optional) 1 mM MgCl2 1 mM DTT. KRas G12D mutant protein was expressed as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent