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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
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Target
Kappa-type opioid receptor
(Human)
The Regents of The University of California
US Patent
Ligand
BDBM579543
(US11484525, Compound DD-144-ANTAGONIST-Covalent)
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Affinity Data
Ki: 0.930nM
Assay Description:
Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Mu-type opioid receptor [N127C]
(Human)
The Regents of The University of California
US Patent
Ligand
BDBM579543
(US11484525, Compound DD-144-ANTAGONIST-Covalent)
Copy SMILES
Copy InChI
Affinity Data
Ki: 18nM
Assay Description:
Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Delta-type opioid receptor
(Human)
The Regents of The University of California
US Patent
Ligand
BDBM579543
(US11484525, Compound DD-144-ANTAGONIST-Covalent)
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Copy InChI
Affinity Data
Ki: 150nM
Assay Description:
Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Kappa-type opioid receptor
(Human)
The Regents of The University of California
US Patent
Ligand
BDBM579543
(US11484525, Compound DD-144-ANTAGONIST-Covalent)
Copy SMILES
Copy InChI
Affinity Data
Ki: 200nM
Assay Description:
Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI