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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMu-type opioid receptor [N127C](Human)
The Regents of The University of California

US Patent
LigandPNGBDBM579564(US11484525, Compound DD-137)
Affinity DataKi:  2.30E+3nMAssay Description:Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetKappa-type opioid receptor(Human)
The Regents of The University of California

US Patent
LigandPNGBDBM579564(US11484525, Compound DD-137)
Affinity DataKi:  8.20E+3nMAssay Description:Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetDelta-type opioid receptor(Human)
The Regents of The University of California

US Patent
LigandPNGBDBM579564(US11484525, Compound DD-137)
Affinity DataKi:  3.60E+4nMAssay Description:Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent