Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 4 hits in this display
IC50: >1.00E+4nMAssay Description:Inhibition of PI3Kalpha in rat Rat1 cells reduction in phosphorylation of AKT at Ser473 residue incubated for 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) incubated for 90 mins by [gamma-33P]-ATP based scintillation counting methodMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of PI3Kalpha (unknown origin) incubated for 90 mins by [gamma-33P]-ATP based scintillation counting methodMore data for this Ligand-Target Pair