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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Gsk

LigandPNGBDBM27848(4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidine, 34 | ...)
Affinity DataIC50:  25nMAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed