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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
37
hits in this display
Target
5-hydroxytryptamine receptor 4
(Guinea pig)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: 5.20nM
Assay Description:
Displacement of [3H]GR-113808 from 5HT4 receptor in guinea pig striatum
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Target
5-hydroxytryptamine receptor 4
(Mouse)
Cnrs Upr 9023
Curated by
PDSP K
i
Database
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: 7.41nM
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Target
5-hydroxytryptamine receptor 4
(Mouse)
Cnrs Upr 9023
Curated by
PDSP K
i
Database
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: 7.94nM
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Target
5-hydroxytryptamine receptor 4
(Mouse)
Cnrs Upr 9023
Curated by
PDSP K
i
Database
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: 7.94nM
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Target
5-hydroxytryptamine receptor 4
(Guinea pig)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: 21nM
Assay Description:
Inhibition of [3H]GR-113808 binding to guinea pig striatum 5-hydroxytryptamine 4 receptor
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Target
5-hydroxytryptamine receptor 4
(Mouse)
Cnrs Upr 9023
Curated by
PDSP K
i
Database
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: 50.1nM
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Target
5-hydroxytryptamine receptor 3A/3B
(Rat)
Searle Research and Development
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: 152nM
Assay Description:
Inhibition of [3H]GR-65630 binding to 5-hydroxytryptamine 3 receptor
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Target
5-hydroxytryptamine receptor 3A/3B
(Rat)
Searle Research and Development
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: 152nM
Assay Description:
Displacement of [3H]GR65630 from 5HT3 receptor in brain cortex from Wistar rat
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Target
5-hydroxytryptamine receptor 3A/3B
(Rat)
Searle Research and Development
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: 152nM
Assay Description:
Inhibition of [3H]GR-65630 binding to rat cortical membrane serotonin 5-hydroxytryptamine 3 receptor
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Target
5-hydroxytryptamine receptor 3A
(Human)
Paris-Sud University
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: 152nM
Assay Description:
Compound was tested for 5-hydroxytryptamine 3 receptor binding affinity
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Target
D(2) dopamine receptor
(Human)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Compound was evaluated for Dopamine receptor D2 binding
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Target
Beta-1/Beta-2/Beta-3 adrenergic receptor
(Rat)
Searle Research and Development
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
The ability to inhibit [3H]dihydroalprenolol prenolol binding to Beta adrenergic receptor in rat whole brain
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Target
5-hydroxytryptamine receptor 1A/1B/1D/1F
(Rat)
Searle Research and Development
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
The ability to inhibit [3H]5-HT binding to 5-hydroxytryptamine 1 receptor in rat cortex
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Target
Serotonin 2 (5-HT2) receptor
(Rat)
Searle Research and Development
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
The ability to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat whole brain
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Target
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(Rat)
Searle Research and Development
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of [3H]GR-65630 binding to 5-hydroxytryptamine 3 receptor
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Target
D(1A) dopamine receptor
(Human)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Compound was evaluated for Dopamine receptor D1 binding
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Target
D(2) dopamine receptor
(Rat)
Dainippon Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Affinity of compound towards Dopamine receptor D2 in rat striatum using [3H]spiperone as radioligand
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Target
D(2) dopamine receptor
(Rat)
Dainippon Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
The ability to inhibit [3H]domperidone binding to dopamine receptor D2 in rat striata
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Target
Alpha-1A adrenergic receptor
(Rat)
Searle Research and Development
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
The ability to inhibit [3H]prazosin binding to Alpha-1 adrenergic receptor in rat whole brain
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Target
D(1A) dopamine receptor
(Rat)
Searle Research and Development
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
The ability to inhibit [3H]-SCH- 23390 binding to Dopamine receptor D1 in rat striata
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Target
Alpha-2A/Alpha-2B/Alpha-2C adrenergic receptor
(Human)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Compound was evaluated for alpha-2 adrenergic receptor binding
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Target
Serotonin 2 (5-HT2) receptor
(Human)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Compound was evaluated for 5-hydroxytryptamine 2 receptor binding
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Target
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Human)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Compound was tested for agonist activity at the 5-hydroxytryptamine 4 receptor in the rat tunica muscularis mucosae (TMM) assay
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Target
5-hydroxytryptamine receptor 1A/1B/1D/1F
(Rat)
Searle Research and Development
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Compound was evaluated for 5-hydroxytryptamine 3 receptor binding
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Target
Beta-1/Beta-2/Beta-3 adrenergic receptor
(Human)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Compound was evaluated for Beta adrenergic receptor binding
More data for this Ligand-Target Pair
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NCI pathway
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Target
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Human)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Binding affinity to adrenergic alpha-1 receptor
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Target
D(2) dopamine receptor
(Human)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Binding affinity to dopamine receptor D2
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Target
D(1A) dopamine receptor
(Human)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Binding affinity to dopamine receptor D1
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Target
Beta-2 adrenergic receptor
(Human)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Binding affinity to adrenergic beta-2 receptor
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Target
Alpha-2A/Alpha-2B/Alpha-2C adrenergic receptor
(Human)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Binding affinity to adrenergic alpha-2 receptor
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Target
Serotonin 2 (5-HT2) receptor
(Human)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Binding affinity to 5HT2 receptor
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Target
Beta-1 adrenergic receptor
(Human)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Binding affinity to adrenergic beta-1 receptor
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Target
5-hydroxytryptamine receptor 4
(Rat)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
EC50: 17nM
Assay Description:
Agonism at 5HT4 receptor in rat tunica muscularis mucosa
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Target
5-hydroxytryptamine receptor 4
(Rat)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
EC50: 23.7nM
Assay Description:
Efficient 5-hydroxytryptamine 4 agonist in the rat tunica muscularis mucosae
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Target
5-hydroxytryptamine receptor 4
(Human)
TBA
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
EC50: 20nM
Assay Description:
Agonist activity against 5-HT4 receptor in rat esophageal muscularis mucosae
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Target
5-hydroxytryptamine receptor 4
(Rat)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Affinity Data
EC50: 66nM
Assay Description:
Tested for agonist activity at the 5-hydroxytryptamine 4 receptor in the rat tunica muscularis mucosae (TMM) assay of racemate mixture
More data for this Ligand-Target Pair
Target Info
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Ligand Info
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In Depth
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Article
PubMed
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Target
5-hydroxytryptamine receptor 4
(Rat)
Pfizer
Curated by
ChEMBL
Ligand
BDBM50005833
((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
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Copy InChI
Affinity Data
EC50: 23nM
Assay Description:
Compound was tested for agonist activity at the 5-hydroxytryptamine 4 receptor in the rat tunica muscularis mucosae (TMM) assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI