Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 24 hits in this display   

TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  1.21E+3nMAssay Description:Inhibition of recombinant ARK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of recombinant VEGFR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  1.83E+3nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  2.22E+3nMAssay Description:Inhibition of recombinant VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  2.87E+3nMAssay Description:Inhibition of recombinant SAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  3.15E+3nMAssay Description:Inhibition of recombinant IGF1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  3.81E+3nMAssay Description:Inhibition of recombinant EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  3.81E+3nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of recombinant INSRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  4.85E+3nMAssay Description:Inhibition of recombinant TIE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  4.85E+3nMAssay Description:Inhibition of recombinant SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of recombinant B-RAF-V600E mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of recombinant Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  5.89E+3nMAssay Description:Inhibition of recombinant CDK4/CycD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  5.89E+3nMAssay Description:Inhibition of recombinant METMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  6.24E+3nMAssay Description:Inhibition of recombinant PDGFRbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  7.28E+3nMAssay Description:Inhibition of recombinant EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  7.97E+3nMAssay Description:Inhibition of recombinant COTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  8.32E+3nMAssay Description:Inhibition of recombinant CDK2/CycAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  9.36E+3nMAssay Description:Inhibition of recombinant ERBB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  1.69E+4nMAssay Description:Inhibition of recombinant FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  1.83E+4nMAssay Description:Inhibition of recombinant AKT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  1.97E+4nMAssay Description:Inhibition of recombinant PLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50: >3.46E+4nMAssay Description:Inhibition of recombinant CK2alpha1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed