Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Gsk

LigandPNGBDBM27805(2-fluoro-6-{[2-({1-[2-(1H-imidazol-1-yl)acetyl]-5-...)
Affinity DataIC50:  32nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Gsk

LigandPNGBDBM27805(2-fluoro-6-{[2-({1-[2-(1H-imidazol-1-yl)acetyl]-5-...)
Affinity DataIC50:  631nMAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing substrate GST-biotin-C-JUN, ATP, and purified activated JNK1alpha1 i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed