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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

Target5-hydroxytryptamine receptor 2A(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50136492(6-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline | 6...)
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity for rat 5-hydroxytryptamine 2A receptor using [3H]-DOBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50136492(6-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline | 6...)
Affinity DataKi:  2.19E+3nMAssay Description:Binding affinity towards cloned rat 5-hydroxytryptamine 2C receptor from fundus tissue by [3H]-mesulergine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50136492(6-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline | 6...)
Affinity DataKi:  4.78E+3nMAssay Description:Binding affinity towards cloned rat 5-hydroxytryptamine 2A receptor by [3H]ketanserin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136492(6-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline | 6...)
Affinity DataKi:  7.83E+3nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Human)
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50136492(6-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline | 6...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of AChEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Human)
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50136492(6-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline | 6...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of BChEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electric eel)
Naresuan University

Curated by ChEMBL
LigandPNGBDBM50136492(6-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline | 6...)
Affinity DataIC50:  2.27E+5nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate measured every 5 sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotase(Bacillus anthracis)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50136492(6-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline | 6...)
Affinity DataKd:  6.75E+5nMAssay Description:Binding affinity to Bacillus anthracis Sterne His-tagged DHOase expressed in Escherichia coli BL21(DE3) Gold cells in presence of N-carbamyl-L-aspart...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotase(Bacillus anthracis)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50136492(6-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline | 6...)
Affinity DataKd:  5.88E+5nMAssay Description:Binding affinity to Bacillus anthracis Sterne His-tagged DHOase expressed in Escherichia coli BL21(DE3) Gold cells by surface plasmon resonance analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed