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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 12 hits in this display   

TargetMitogen-activated protein kinase kinase kinase 20(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50513866(CHEMBL4450810)
Affinity DataIC50:  4nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human full-length ZAK expressed in baculovirus infected Sf9 insect cells using MBP as substrate after...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50513866(CHEMBL4450810)
Affinity DataIC50:  156nMAssay Description:Inhibition of human ABL1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50513866(CHEMBL4450810)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human B-RAF V600E mutant using Ser/Thr3 as substrate after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLIM domain kinase 1(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50513866(CHEMBL4450810)
Affinity DataKd:  23nMAssay Description:Binding affinity to human LIMK1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50513866(CHEMBL4450810)
Affinity DataKd:  63nMAssay Description:Binding affinity to human LIMK2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50513866(CHEMBL4450810)
Affinity DataKd:  160nMAssay Description:Binding affinity to human LCKMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 20(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50513866(CHEMBL4450810)
Affinity DataKd:  8nMAssay Description:Binding affinity to ATP-binding site of human ZAK expressed in Escherichia coli by active site-dependent competition binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50513866(CHEMBL4450810)
Affinity DataKd:  530nMAssay Description:Binding affinity to human FLT3 F691L mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50513866(CHEMBL4450810)
Affinity DataKd:  190nMAssay Description:Binding affinity to human BLKMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50513866(CHEMBL4450810)
Affinity DataKd:  15nMAssay Description:Binding affinity to human ABL1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 20(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50513866(CHEMBL4450810)
Affinity DataKd:  8nMAssay Description:Binding affinity to human ZAKMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50513866(CHEMBL4450810)
Affinity DataKd:  57nMAssay Description:Binding affinity to human RIPK2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed