Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rat)
Pfizer

Curated by ChEMBL

LigandBDBM50222052(CHEMBL329548)Copy SMILESCopy InChI

Affinity DataKi:  6.20nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

Target5-hydroxytryptamine receptor 7(Rat)
Pfizer

Curated by ChEMBL

LigandBDBM50222052(CHEMBL329548)Copy SMILESCopy InChI

Affinity DataKi:  17nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Pfizer

Curated by ChEMBL

LigandBDBM50222052(CHEMBL329548)Copy SMILESCopy InChI

Affinity DataKi:  102nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI