Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University of Nebraska Medical Center

Curated by ChEMBL

LigandBDBM50532048(CHEMBL4536665)Copy SMILESCopy InChI

Affinity DataEC50:  183nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetG protein-activated inward rectifier potassium channel 4(Homo sapiens (Human))
University of Nebraska Medical Center

Curated by ChEMBL

LigandBDBM50532048(CHEMBL4536665)Copy SMILESCopy InChI

Affinity DataEC50:  619nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair

Target InfoReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI