Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 12 hits in this display
BDBM185590(US9156852, 105 | USRE47451, Example 105)
BDBM185590(US9156852, 105 | USRE47451, Example 105)
BDBM185590(US9156852, 105 | USRE47451, Example 105)
IC50: 31nMAssay Description:The compounds prepared in Examples were tested for inhibitory activity against three subtypes of RAF, i.e., RAF1 Y340D Y341D (C-RAF), B-RAF normal ty...More data for this Ligand-Target Pair
BDBM185590(US9156852, 105 | USRE47451, Example 105)
IC50: 31nMAssay Description:The compounds prepared in Examples were tested for inhibitory activity against three subtypes of RAF, i.e., RAF1 Y340D Y341D (C-RAF), B-RAF normal ty...More data for this Ligand-Target Pair
BDBM185590(US9156852, 105 | USRE47451, Example 105)
BDBM185590(US9156852, 105 | USRE47451, Example 105)
BDBM185590(US9156852, 105 | USRE47451, Example 105)
IC50: 71nMAssay Description:As such, the compounds prepared in Examples were tested for inhibitory activity against FMS, DDR1 and DDR2 kinases using Kinase Screening and Profili...More data for this Ligand-Target Pair
BDBM185590(US9156852, 105 | USRE47451, Example 105)
IC50: 71nMAssay Description:The compounds prepared in Examples were tested for inhibitory activity against FMS, DDR1 and DDR2 kinases using Kinase Screening and Profiling Servic...More data for this Ligand-Target Pair
BDBM185590(US9156852, 105 | USRE47451, Example 105)
IC50: 179nMAssay Description:The compounds prepared in Examples were tested for inhibitory activity against three subtypes of RAF, i.e., RAF1 Y340D Y341D (C-RAF), B-RAF normal ty...More data for this Ligand-Target Pair
BDBM185590(US9156852, 105 | USRE47451, Example 105)
IC50: 179nMAssay Description:The compounds prepared in Examples were tested for inhibitory activity against three subtypes of RAF, i.e., RAF1 Y340D Y341D (C-RAF), B-RAF normal ty...More data for this Ligand-Target Pair
BDBM185590(US9156852, 105 | USRE47451, Example 105)
IC50: 181nMAssay Description:As such, the compounds prepared in Examples were tested for inhibitory activity against FMS, DDR1 and DDR2 kinases using Kinase Screening and Profili...More data for this Ligand-Target Pair
BDBM185590(US9156852, 105 | USRE47451, Example 105)
IC50: 181nMAssay Description:The compounds prepared in Examples were tested for inhibitory activity against FMS, DDR1 and DDR2 kinases using Kinase Screening and Profiling Servic...More data for this Ligand-Target Pair