Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 7 hits in this display
BDBM364535(Cis 3-[6-(1,3-Dimethyl-1H-pyrazol-4-yl)-pyrazin-2-...)
BDBM364535(Cis 3-[6-(1,3-Dimethyl-1H-pyrazol-4-yl)-pyrazin-2-...)
BDBM364535(Cis 3-[6-(1,3-Dimethyl-1H-pyrazol-4-yl)-pyrazin-2-...)
IC50: 100nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
BDBM364535(Cis 3-[6-(1,3-Dimethyl-1H-pyrazol-4-yl)-pyrazin-2-...)
IC50: 630nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta™ Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, U...More data for this Ligand-Target Pair
BDBM364535(Cis 3-[6-(1,3-Dimethyl-1H-pyrazol-4-yl)-pyrazin-2-...)
IC50: 4.40E+3nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
BDBM364535(Cis 3-[6-(1,3-Dimethyl-1H-pyrazol-4-yl)-pyrazin-2-...)
BDBM364535(Cis 3-[6-(1,3-Dimethyl-1H-pyrazol-4-yl)-pyrazin-2-...)
IC50: >1.00E+4nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair