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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Nuclear receptor subfamily 4 group A member 1
(Human)
Burnham Center For Chemical Genomics
Curated by
PubChem BioAssay
Ligand
BDBM40571
(3-amino-6-methyl-7-thiazolo[3,2-b][1,2,4]triazinon...)
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Affinity Data
IC50: >1.25E+4nM
Assay Description:
Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (San Diego, CA) NIH Molecular Libraries Screening Cen...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
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PC sid
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PCBioAssay
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Target
Mitogen-activated protein kinase kinase kinase kinase 2
(Human)
Nmmlsc
Curated by
PubChem BioAssay
Ligand
BDBM40571
(3-amino-6-methyl-7-thiazolo[3,2-b][1,2,4]triazinon...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 4.09E+3nM
Assay Description:
University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...
More data for this Ligand-Target Pair
Target Info
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Patents
In Depth
Details
PCBioAssay
Copy BDB DOI
Target
Mitogen-activated protein kinase kinase kinase kinase 2
(Human)
Nmmlsc
Curated by
PubChem BioAssay
Ligand
BDBM40571
(3-amino-6-methyl-7-thiazolo[3,2-b][1,2,4]triazinon...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 3.40E+3nM
Assay Description:
University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...
More data for this Ligand-Target Pair
Target Info
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Patents
In Depth
Details
PCBioAssay
Copy BDB DOI