Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 7 hits in this display
BDBM295128(3-(6-Amino-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridi...)
BDBM295128(3-(6-Amino-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridi...)
IC50: 160nMpH: 7.5Assay Description:The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad, Calif., USA) (Cat. No. PV5099). The kit contains t...More data for this Ligand-Target Pair
BDBM295128(3-(6-Amino-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridi...)
BDBM295128(3-(6-Amino-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridi...)
IC50: 3.90E+3nMpH: 7.5 T: 2°CAssay Description:The luminescence-based ATP detection reagent KinaseGlo was obtained from Promega, (Cat. No. V6714, Lot No. 236161) through Catalys, Wallisellen, Swit...More data for this Ligand-Target Pair
BDBM295128(3-(6-Amino-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridi...)
IC50: 5.40E+3nMpH: 7.5 T: 2°CAssay Description:The luminescence-based ATP detection reagent KinaseGlo was obtained from Promega, (Cat. No. V6714, Lot No. 236161) through Catalys, Wallisellen, Swit...More data for this Ligand-Target Pair
BDBM295128(3-(6-Amino-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridi...)
IC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:The luminescence-based ATP detection reagent KinaseGlo was obtained from Promega, (Cat. No. V6714, Lot No. 236161) through Catalys, Wallisellen, Swit...More data for this Ligand-Target Pair
BDBM295128(3-(6-Amino-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridi...)