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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

LigandPNGBDBM50228627(CHEMBL1203566)
Affinity DataKi:  19nMAssay Description:Binding affinity was determined against alpha-2 adrenergic receptor of rat cerebral cortex using [3H]yohimbine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228627(CHEMBL1203566)
Affinity DataKi:  95nMAssay Description:Binding affinity was determined against alpha-2 adrenergic receptor of rat cerebral cortex using [3H]idazoxan as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50228627(CHEMBL1203566)
Affinity DataKi:  6.46E+3nMAssay Description:Binding affinity determined to alpha-1 adrenergic receptor of rat cerebral cortex using [3H]prazosin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed