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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
1
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Target
Chloroquine resistance transporter
(malaria parasite P. falciparum)
University of Siena
Curated by
ChEMBL
Ligand
BDBM50396334
(CHEMBL2170034)
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Affinity Data
IC50: 1.03E+4nM
Assay Description:
Inhibition of chloroquine-resistant Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocyte assessed as inhibition of [3H]chloroquine uptake...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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