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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
1
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Target
NACHT, LRR and PYD domains-containing protein 3
(Human)
Jecure Therapeutics
Curated by
ChEMBL
Ligand
BDBM50607500
(CHEMBL5220827)
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Affinity Data
IC50: 2.55E+3nM
Assay Description:
Inhibition of NLRP3 inflammasome activation in LPS and nigericin-stimulated human PBMC cells assessed as reduction in IL-1beta release preincubated w...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
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