Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 18 hits in this display
BDBM569273(US11427563, Compound 14 | US11427563, Compound 157...)
BDBM569273(US11427563, Compound 14 | US11427563, Compound 157...)
IC50: 0.900nMAssay Description:Compounds were prepared in the exact same manner as described in the ROCK Kinase Assay with the exception to the substrate and enzyme. The JAK 2× sub...More data for this Ligand-Target Pair
BDBM569273(US11427563, Compound 14 | US11427563, Compound 157...)
IC50: 0.900nMAssay Description:Compounds were prepared in the exact same manner as described in the ROCK Kinase Assay with the exception to the substrate and enzyme. The JAK 2× sub...More data for this Ligand-Target Pair
BDBM569273(US11427563, Compound 14 | US11427563, Compound 157...)
IC50: 9nMAssay Description:Compounds were prepared in the exact same manner as described in the ROCK Kinase Assay with the exception to the substrate and enzyme. The JAK 2× sub...More data for this Ligand-Target Pair
BDBM569273(US11427563, Compound 14 | US11427563, Compound 157...)
IC50: 9nMAssay Description:Compounds were prepared in the exact same manner as described in the ROCK Kinase Assay with the exception to the substrate and enzyme. The JAK 2× sub...More data for this Ligand-Target Pair
BDBM569273(US11427563, Compound 14 | US11427563, Compound 157...)
IC50: 9nMAssay Description:Compounds were prepared in the exact same manner as described in the ROCK Kinase Assay with the exception to the substrate and enzyme. The JAK 2× sub...More data for this Ligand-Target Pair
BDBM569273(US11427563, Compound 14 | US11427563, Compound 157...)
IC50: 11nMAssay Description:Compounds were prepared in the exact same manner as described in the ROCK Kinase Assay with the exception to the substrate and enzyme. The JAK 2× sub...More data for this Ligand-Target Pair
BDBM569273(US11427563, Compound 14 | US11427563, Compound 157...)
IC50: 12.5nMAssay Description:Compounds were prepared in the exact same manner as described in the ROCK Kinase Assay with the exception to the substrate and enzyme. The JAK 2× sub...More data for this Ligand-Target Pair
BDBM569273(US11427563, Compound 14 | US11427563, Compound 157...)
BDBM569273(US11427563, Compound 14 | US11427563, Compound 157...)
IC50: 16nMAssay Description:All compounds were initially prepared as 10 mM stocks in anhydrous dimethylsulfoxide (DMSO). A 20 μl aliquot of the 10 mM solutions was transfer...More data for this Ligand-Target Pair
BDBM569273(US11427563, Compound 14 | US11427563, Compound 157...)
IC50: 16nMAssay Description:All compounds were initially prepared as 10 mM stocks in anhydrous dimethylsulfoxide (DMSO). A 20 μl aliquot of the 10 mM solutions was transfer...More data for this Ligand-Target Pair
BDBM569273(US11427563, Compound 14 | US11427563, Compound 157...)
IC50: 108nMAssay Description:All compounds were initially prepared as 10 mM stocks in anhydrous dimethylsulfoxide (DMSO). A 20 μl aliquot of the 10 mM solutions was transfer...More data for this Ligand-Target Pair
BDBM569273(US11427563, Compound 14 | US11427563, Compound 157...)
IC50: 108nMAssay Description:All compounds were initially prepared as 10 mM stocks in anhydrous dimethylsulfoxide (DMSO). A 20 μl aliquot of the 10 mM solutions was transfer...More data for this Ligand-Target Pair
BDBM569273(US11427563, Compound 14 | US11427563, Compound 157...)
IC50: 108nMAssay Description:All compounds were initially prepared as 10 mM stocks in anhydrous dimethylsulfoxide (DMSO). A 20 μl aliquot of the 10 mM solutions was transfer...More data for this Ligand-Target Pair
BDBM569273(US11427563, Compound 14 | US11427563, Compound 157...)
IC50: 122nMAssay Description:All compounds were initially prepared as 10 mM stocks in anhydrous dimethylsulfoxide (DMSO). A 20 μl aliquot of the 10 mM solutions was transfer...More data for this Ligand-Target Pair
BDBM569273(US11427563, Compound 14 | US11427563, Compound 157...)
IC50: 122nMAssay Description:All compounds were initially prepared as 10 mM stocks in anhydrous dimethylsulfoxide (DMSO). A 20 μl aliquot of the 10 mM solutions was transfer...More data for this Ligand-Target Pair
BDBM569273(US11427563, Compound 14 | US11427563, Compound 157...)
IC50: 122nMAssay Description:All compounds were initially prepared as 10 mM stocks in anhydrous dimethylsulfoxide (DMSO). A 20 μl aliquot of the 10 mM solutions was transfer...More data for this Ligand-Target Pair
BDBM569273(US11427563, Compound 14 | US11427563, Compound 157...)
IC50: 200nMAssay Description:All compounds were initially prepared as 10 mM stocks in anhydrous dimethylsulfoxide (DMSO). A 20 μl aliquot of the 10 mM solutions was transfer...More data for this Ligand-Target Pair