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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
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Target
Transitional endoplasmic reticulum ATPase
(Human)
Kyowa Hakko Kogyo
Curated by
ChEMBL
Ligand
BDBM50312873
(4-(4-(pyridin-2-yl)thiazol-2-ylamino)phenol | 4-{[...)
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Affinity Data
IC50: 230nM
Assay Description:
Inhibition of VCP assessed as conversion of ATP to ADP by enzyme coupled glucokinase assay
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Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
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Article
PubMed
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Target
Nuclear receptor subfamily 4 group A member 1
(Human)
Sanford-Burnham Center For Chemical Genomics
Curated by
PubChem BioAssay
Ligand
BDBM50312873
(4-(4-(pyridin-2-yl)thiazol-2-ylamino)phenol | 4-{[...)
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Affinity Data
EC50: 3.69E+3nM
Assay Description:
Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
PCBioAssay
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