Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMenin(Homo sapiens (Human))
TBA

Curated by ChEMBL

LigandBDBM50511899(CHEMBL4457657 | US11045448, Cpd. No. 67)Copy SMILESCopy InChI

Affinity DataIC50:  1.70nMAssay Description:Inhibition of fluorescent labeled tracer binding to Menin (unknown origin) after 1 hr by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetMenin(Homo sapiens (Human))
TBA

Curated by ChEMBL

LigandBDBM50511899(CHEMBL4457657 | US11045448, Cpd. No. 67)Copy SMILESCopy InChI

Affinity DataIC50:  2nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI