Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetTissue factor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

LigandBDBM50235153(CHEBI:67985 | CHEMBL510111)Copy SMILESCopy InChI

Affinity DataIC50:  0.0350nMAssay Description:Inhibition of LPS-induced tissue factor procoagulant activity in human THP1 cells preincubated for 1 hr followed by LPS addition measured after 5 hrs...More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPurchaseCHEMBLKEGGPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
China Pharmaceutical University

LigandBDBM23204((2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl...)Copy SMILESCopy InChI

Affinity DataIC50:  2.93E+5nMpH: 7.2 T: 2°CAssay Description:The activity of the compounds is determined by measuring the inhibitory effect of the compounds in the direction of glycogen synthesis, the conversio...More data for this Ligand-Target Pair

Target InfoPDBMMDBKEGG
UniProtKB/SwissProt
B.MOADDrugBankGoogleScholar

Ligand InfoPurchaseKEGGPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI