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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetPotassium voltage-gated channel subfamily A member 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50115814(CHEMBL3609062)
Affinity DataIC50:  0.00300nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50115814(CHEMBL3609062)
Affinity DataIC50:  0.0360nMAssay Description:Antagonist activity at Kv1.3 in human whole blood assessed as inhibition of thapsigargin-induced IL-2 secretion incubated for 30 prior to thapsigargi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50115814(CHEMBL3609062)
Affinity DataIC50:  0.0730nMAssay Description:Antagonist activity at Kv1.3 in human whole blood assessed as inhibition of thapsigargin-induced IFN-gamma secretion incubated for 30 prior to thapsi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50115814(CHEMBL3609062)
Affinity DataIC50:  0.154nMAssay Description:Antagonist activity at human Kv1.3 expressed in CHOK1 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch clam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed