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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50124406(CHEMBL3623450)
Affinity DataKd:  6.57E+3nMAssay Description:Binding affinity to GST-tagged Grb7-SH2 domain (415 to 532 amino acid residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using 50 mM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 10(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50124406(CHEMBL3623450)
Affinity DataKd:  4.20E+5nMAssay Description:Binding affinity to GST-tagged Grb10-SH2 domain (471 to 594 amino acid residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using 20 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50124406(CHEMBL3623450)
Affinity DataKd:  5.60E+5nMAssay Description:Binding affinity to GST-tagged Grb2-SH2 domain (58 to 160 amino acid residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using 20 mM ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50124406(CHEMBL3623450)
Affinity DataKd:  2.10E+3nMAssay Description:Binding affinity to GST-tagged Grb7-SH2 domain (415 to 532 amino acid residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using 20 mM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed