Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 16 hits in this display
BDBM50241487(2,3,6,23-tetrahydroxyurs-12-en-28-oic acid | Asiat...)
BDBM23202((1S,2R,4aS,6aS,6bR,9R,10R,11R,12aR,12bR,14bS)-10,1...)
BDBM50241487(2,3,6,23-tetrahydroxyurs-12-en-28-oic acid | Asiat...)
BDBM50241487(2,3,6,23-tetrahydroxyurs-12-en-28-oic acid | Asiat...)
BDBM50241487(2,3,6,23-tetrahydroxyurs-12-en-28-oic acid | Asiat...)
BDBM50241487(2,3,6,23-tetrahydroxyurs-12-en-28-oic acid | Asiat...)
BDBM50241487(2,3,6,23-tetrahydroxyurs-12-en-28-oic acid | Asiat...)
BDBM50241487(2,3,6,23-tetrahydroxyurs-12-en-28-oic acid | Asiat...)
BDBM50241487(2,3,6,23-tetrahydroxyurs-12-en-28-oic acid | Asiat...)
BDBM50241487(2,3,6,23-tetrahydroxyurs-12-en-28-oic acid | Asiat...)
IC50: >4.00E+4nMAssay Description:Inhibition of ovine recombinant COX1 assessed as decrease in formation of PGE2 using arachidonic acid as substrate preincubated for 10 mins followed ...More data for this Ligand-Target Pair
BDBM50241487(2,3,6,23-tetrahydroxyurs-12-en-28-oic acid | Asiat...)
IC50: >4.00E+4nMAssay Description:Inhibition of human recombinant 5-LOX expressed in insect cells assessed as decrease in production of 5-HPETE and 5-HETE using arachidonic acid as su...More data for this Ligand-Target Pair
BDBM50241487(2,3,6,23-tetrahydroxyurs-12-en-28-oic acid | Asiat...)
IC50: >4.00E+4nMAssay Description:Inhibition of human recombinant COX2 expressed in baculovirus infected sf21 cells assessed as decrease in PGE2 formation using arachidonic acid as su...More data for this Ligand-Target Pair
BDBM50241487(2,3,6,23-tetrahydroxyurs-12-en-28-oic acid | Asiat...)
BDBM50241487(2,3,6,23-tetrahydroxyurs-12-en-28-oic acid | Asiat...)
BDBM50241487(2,3,6,23-tetrahydroxyurs-12-en-28-oic acid | Asiat...)
BDBM50241487(2,3,6,23-tetrahydroxyurs-12-en-28-oic acid | Asiat...)