Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetRAC-alpha/RAC-beta/RAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50550738(CHEMBL4792262)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human AKT assessed as inhibition of substrate phosphorylation using AKTide-2T as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50550738(CHEMBL4792262)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of MMP-9 (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50550738(CHEMBL4792262)
Affinity DataIC50:  104nMAssay Description:Inhibition of MMP-1 (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50550738(CHEMBL4792262)
Affinity DataIC50:  266nMAssay Description:Inhibition of MMP-2 (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50550738(CHEMBL4792262)
Affinity DataIC50:  280nMAssay Description:Inhibition of MMP-13 (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed