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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Cystic fibrosis transmembrane conductance regulator
(Homo sapiens (Human))
University Of California
Curated by
ChEMBL
Ligand
BDBM50237256
(CHEMBL4068723)
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Affinity Data
EC50: 21nM
Assay Description:
Activation of human CFTR expressed in forskolin-stimulated basolateral membrane permeabilized FRT cells assessed as increase in short-circuit current...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Cystic fibrosis transmembrane conductance regulator
(Homo sapiens (Human))
University Of California
Curated by
ChEMBL
Ligand
BDBM50237256
(CHEMBL4068723)
Copy SMILES
Copy InChI
Affinity Data
EC50: 21nM
Assay Description:
Potentiation of CFTR in FRT cells co-expressing human wild-type CFTR and YFP iodide-sensing protein in presence of forskolin measured by High-Through...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Cystic fibrosis transmembrane conductance regulator
(Homo sapiens (Human))
University Of California
Curated by
ChEMBL
Ligand
BDBM50237256
(CHEMBL4068723)
Copy SMILES
Copy InChI
Affinity Data
EC50: 9nM
Assay Description:
In vitro inhibition of farnesyl-protein transferase
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI