Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50237256(CHEMBL4068723)
Affinity DataEC50:  21nMAssay Description:Activation of human CFTR expressed in forskolin-stimulated basolateral membrane permeabilized FRT cells assessed as increase in short-circuit current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50237256(CHEMBL4068723)
Affinity DataEC50:  21nMAssay Description:Potentiation of CFTR in FRT cells co-expressing human wild-type CFTR and YFP iodide-sensing protein in presence of forskolin measured by High-Through...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50237256(CHEMBL4068723)
Affinity DataEC50:  9nMAssay Description:In vitro inhibition of farnesyl-protein transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed