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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
9
hits in this display
Target
Collagenase 3
(Homo sapiens (Human))
Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50233887
(CHEMBL1511860)
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Affinity Data
IC50: 1.90E+3nM
Assay Description:
Inhibition of APMA-activated recombinant human MMP-13 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
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PubMed
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Target
Matrix metalloproteinase-9
(Homo sapiens (Human))
Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50233887
(CHEMBL1511860)
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Affinity Data
IC50: 2.20E+3nM
Assay Description:
Inhibition of APMA-activated recombinant human MMP-9 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric m...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
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PC sid
Patents
In Depth
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Article
PubMed
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Target
72 kDa type IV collagenase
(Homo sapiens (Human))
Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50233887
(CHEMBL1511860)
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Affinity Data
IC50: 3.60E+3nM
Assay Description:
Inhibition of APMA-activated recombinant human MMP-2 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric m...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
PC cid
PC sid
Patents
In Depth
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Article
PubMed
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Target
Matrix metalloproteinase-14
(Homo sapiens (Human))
Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50233887
(CHEMBL1511860)
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Affinity Data
IC50: 7.50E+3nM
Assay Description:
Inhibition of APMA-activated recombinant human GST-tagged MMP-14 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofl...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
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PC sid
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In Depth
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Article
PubMed
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Target
Neutrophil collagenase
(Homo sapiens (Human))
Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50233887
(CHEMBL1511860)
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Affinity Data
IC50: 9.30E+3nM
Assay Description:
Inhibition of APMA-activated recombinant human MMP-8 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric m...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
PC cid
PC sid
Patents
In Depth
Details
Article
PubMed
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Target
Matrilysin
(Homo sapiens (Human))
Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50233887
(CHEMBL1511860)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of APMA-activated recombinant human MMP-7 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric m...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
PC cid
PC sid
Patents
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Interstitial collagenase
(Homo sapiens (Human))
Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50233887
(CHEMBL1511860)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of APMA-activated recombinant human MMP-1 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric m...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
PC cid
PC sid
Patents
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Stromelysin-1
(Homo sapiens (Human))
Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50233887
(CHEMBL1511860)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of APMA-activated recombinant human MMP-3 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric m...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Stromelysin-2
(Homo sapiens (Human))
Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50233887
(CHEMBL1511860)
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Affinity Data
IC50: 8.30E+4nM
Assay Description:
Inhibition of APMA-activated recombinant human MMP-10 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
Article
PubMed
Copy BDB DOI