Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 8 hits in this display
BDBM50337729(CHEMBL1615186 | N-((2S,4S)-1-(4-(2,4-dichlorobenzy...)
BDBM50337729(CHEMBL1615186 | N-((2S,4S)-1-(4-(2,4-dichlorobenzy...)
BDBM50337729(CHEMBL1615186 | N-((2S,4S)-1-(4-(2,4-dichlorobenzy...)
IC50: 3.5nMAssay Description:Protein concentrations were measured using the Micro BCA Protein Assay Kit (Pierce/Thermo Scientific, IL). Sample buffer was mixed with 5-25 μg ...More data for this Ligand-Target Pair
BDBM50337729(CHEMBL1615186 | N-((2S,4S)-1-(4-(2,4-dichlorobenzy...)
BDBM50337729(CHEMBL1615186 | N-((2S,4S)-1-(4-(2,4-dichlorobenzy...)
IC50: 430nMAssay Description:Inhibition of recombinant human MMP14 assessed as substrate cleavage by measuring increase in fluorescence after 16 hrsMore data for this Ligand-Target Pair
BDBM50337729(CHEMBL1615186 | N-((2S,4S)-1-(4-(2,4-dichlorobenzy...)
IC50: 430nMAssay Description:Inhibition of recombinant human MMP13 assessed as substrate cleavage by measuring increase in fluorescence after 16 hrsMore data for this Ligand-Target Pair
BDBM50337729(CHEMBL1615186 | N-((2S,4S)-1-(4-(2,4-dichlorobenzy...)
BDBM50337729(CHEMBL1615186 | N-((2S,4S)-1-(4-(2,4-dichlorobenzy...)
IC50: >1.00E+4nMAssay Description:Inhibition of recombinant human MMP1 assessed as substrate cleavage by measuring increase in fluorescence after 16 hrsMore data for this Ligand-Target Pair