Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetSentrin-specific protease 1(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL

LigandBDBM50346606(CHEMBL1797137)Copy SMILESCopy InChI

Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of recombinant human SENP1 catalytic domain using RanGAP1 as substrate preincubated for 10 mins followed by substrate addition and measure...More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails PubMed
Copy BDB DOI

TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Chinese Academy Of Sciences

Curated by ChEMBL

LigandBDBM50346606(CHEMBL1797137)Copy SMILESCopy InChI

Affinity DataIC50:  1.88E+5nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 mins by microplate reader bas...More data for this Ligand-Target Pair

Target InfoPDBMMDBKEGG
UniProtKB/SwissProt
B.MOADDrugBankGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI