Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 11 hits in this display
BDBM50158595((4'-(3-((2R,5R)-2,5-dimethylpyrrolidin-1-yl)propox...)
BDBM50158595((4'-(3-((2R,5R)-2,5-dimethylpyrrolidin-1-yl)propox...)
BDBM50158595((4'-(3-((2R,5R)-2,5-dimethylpyrrolidin-1-yl)propox...)
BDBM50158595((4'-(3-((2R,5R)-2,5-dimethylpyrrolidin-1-yl)propox...)
BDBM50158595((4'-(3-((2R,5R)-2,5-dimethylpyrrolidin-1-yl)propox...)
BDBM50158595((4'-(3-((2R,5R)-2,5-dimethylpyrrolidin-1-yl)propox...)
BDBM50158595((4'-(3-((2R,5R)-2,5-dimethylpyrrolidin-1-yl)propox...)
Ki: 1.66nMAssay Description:In vitro binding affinity was determined as displacement of [3H]N-R-methylhistamine from C6 cell membranes expressing rat histamine H3 receptorMore data for this Ligand-Target Pair
BDBM50158595((4'-(3-((2R,5R)-2,5-dimethylpyrrolidin-1-yl)propox...)
BDBM50158595((4'-(3-((2R,5R)-2,5-dimethylpyrrolidin-1-yl)propox...)
BDBM50158595((4'-(3-((2R,5R)-2,5-dimethylpyrrolidin-1-yl)propox...)
BDBM50158595((4'-(3-((2R,5R)-2,5-dimethylpyrrolidin-1-yl)propox...)