Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 18 hits in this display
BDBM379697(US9926281, Compound 255)
IC50: 19nMAssay Description:Inhibition of human recombinant ADAMTS-5 assessed as cleavage of fluorescent substrate using FAM-TBIS-1 by biochemical assayMore data for this Ligand-Target Pair
BDBM379697(US9926281, Compound 255)
ADAMTS5(Rattus norvegicus (Rat))Galapagos
US Patent
BDBM379697(US9926281, Compound 255)
BDBM379697(US9926281, Compound 255)
BDBM379697(US9926281, Compound 255)
BDBM379697(US9926281, Compound 255)
BDBM379697(US9926281, Compound 255)
BDBM379697(US9926281, Compound 255)
BDBM379697(US9926281, Compound 255)
BDBM379697(US9926281, Compound 255)
BDBM379697(US9926281, Compound 255)
BDBM379697(US9926281, Compound 255)
BDBM379697(US9926281, Compound 255)
BDBM379697(US9926281, Compound 255)
BDBM379697(US9926281, Compound 255)
BDBM379697(US9926281, Compound 255)
BDBM379697(US9926281, Compound 255)
BDBM379697(US9926281, Compound 255)