Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 12 hits in this display
BDBM50081280(CHEMBL3422005 | US9840508, Compound 2)
Ki: 100nMAssay Description:Displacement of [3H]-SB222200 from recombinant human NK3R expressed in CHO cell membranes after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM50081280(CHEMBL3422005 | US9840508, Compound 2)
BDBM50081280(CHEMBL3422005 | US9840508, Compound 2)
Ki: 100nMAssay Description:The ability of compounds of the invention to inhibit the binding of the NK-3 receptor selective antagonist 3H-SB222200 was assessed by an in vitro ra...More data for this Ligand-Target Pair
BDBM50081280(CHEMBL3422005 | US9840508, Compound 2)
BDBM50081280(CHEMBL3422005 | US9840508, Compound 2)
BDBM50081280(CHEMBL3422005 | US9840508, Compound 2)
BDBM50081280(CHEMBL3422005 | US9840508, Compound 2)
IC50: 160nMAssay Description:The ability of compounds of the invention to inhibit the binding of the NK-3 receptor selective antagonist 3H-SB222200 was assessed by an in vitro ra...More data for this Ligand-Target Pair
BDBM50081280(CHEMBL3422005 | US9840508, Compound 2)
BDBM50081280(CHEMBL3422005 | US9840508, Compound 2)
BDBM50081280(CHEMBL3422005 | US9840508, Compound 2)
BDBM50081280(CHEMBL3422005 | US9840508, Compound 2)
BDBM50081280(CHEMBL3422005 | US9840508, Compound 2)