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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50111696(5-Bromo-2-[(4-but-2-ynyloxy-benzenesulfonyl)-methy...)
Affinity DataIC50:  16nMAssay Description:Inhibition of porcine Tumor necrosis factor alpha converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50111696(5-Bromo-2-[(4-but-2-ynyloxy-benzenesulfonyl)-methy...)
Affinity DataIC50:  16nMAssay Description:Inhibition of Tumor necrosis factor alpha converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50111696(5-Bromo-2-[(4-but-2-ynyloxy-benzenesulfonyl)-methy...)
Affinity DataIC50:  154nMAssay Description:Inhibition of Matrix metalloproteinase-13 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50111696(5-Bromo-2-[(4-but-2-ynyloxy-benzenesulfonyl)-methy...)
Affinity DataIC50:  154nMAssay Description:Inhibition of Matrix metalloproteinase-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50111696(5-Bromo-2-[(4-but-2-ynyloxy-benzenesulfonyl)-methy...)
Affinity DataIC50:  304nMAssay Description:Inhibition of Matrix metalloproteinase-9 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50111696(5-Bromo-2-[(4-but-2-ynyloxy-benzenesulfonyl)-methy...)
Affinity DataIC50:  304nMAssay Description:Inhibition of Matrix metalloproteinase-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50111696(5-Bromo-2-[(4-but-2-ynyloxy-benzenesulfonyl)-methy...)
Affinity DataIC50:  1.62E+3nMAssay Description:Inhibition of Matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50111696(5-Bromo-2-[(4-but-2-ynyloxy-benzenesulfonyl)-methy...)
Affinity DataIC50:  1.62E+3nMAssay Description:Inhibition of Matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed