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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50131523((R)-2-(4-(but-2-ynyloxy)phenylsulfonamido)-N-hydro...)
Affinity DataIC50:  4nMAssay Description:In vitro inhibition of tumor necrosis factor-alpha converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50131523((R)-2-(4-(but-2-ynyloxy)phenylsulfonamido)-N-hydro...)
Affinity DataIC50:  195nMAssay Description:In vitro inhibition of Matrix metalloprotein 13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50131523((R)-2-(4-(but-2-ynyloxy)phenylsulfonamido)-N-hydro...)
Affinity DataIC50:  794nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50131523((R)-2-(4-(but-2-ynyloxy)phenylsulfonamido)-N-hydro...)
Affinity DataIC50:  796nMAssay Description:In vitro inhibition of Matrix metalloprotein-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50131523((R)-2-(4-(but-2-ynyloxy)phenylsulfonamido)-N-hydro...)
Affinity DataIC50:  4.03E+3nMAssay Description:In vitro inhibition of Matrix metalloprotein 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50131523((R)-2-(4-(but-2-ynyloxy)phenylsulfonamido)-N-hydro...)
Affinity DataIC50:  4.07E+3nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed